New thiopyrimidine-benzenesulfonamide conjugates as selective carbonic anhydrase II inhibitors: synthesis, in vitro biological evaluation, and molecular docking studies-Reference-Cited by-同舟云学术

New thiopyrimidine-benzenesulfonamide conjugates as selective carbonic anhydrase II inhibitors: synthesis, in vitro biological evaluation, and molecular docking studies

Published:2020-03 Issue:5 Volume:28 Page:115329
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Abdel-Mohsen Heba T.,El Kerdawy Ahmed M.,Omar Mohamed A.,Berrino Emanuela,Abdelsamie Ahmed S.,El Diwani Hoda I.,Supuran Claudiu T.

Funder

STDF

UCSF

University of California, San Francisco

National Institutes of Health

National Center for Research Resources

National Institute of General Medical Sciences

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference51 articles.

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4. Structural annotation of human carbonic anhydrases;Aggarwal;J Enzym Inhib Med Chem,2013

5. Carbonic anhydrase as a model for biophysical and physical-organic studies of proteins and protein-ligand binding;Krishnamurthy;Chem Rev,2008

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