Novel indolylarylsulfone derivatives as covalent HIV-1 reverse transcriptase inhibitors specifically targeting the drug-resistant mutant Y181C-Reference-Cited by-同舟云学术

Novel indolylarylsulfone derivatives as covalent HIV-1 reverse transcriptase inhibitors specifically targeting the drug-resistant mutant Y181C

Published:2021-01 Issue: Volume:30 Page:115927
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Gao Ping,Song Shu,Frutos-Beltrán Estrella,Li Wenxin,Sun Bin,Kang Dongwei,Zou Jinmi,Zhang Jian,Pannecouque Christophe,De Clercq Erik,Menéndez-Arias Luis,Zhan Peng,Liu Xinyong

Funder

Shandong University

Spanish National Plan for Scientific and Technical Research and Innovation

Government of Shandong Province

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference20 articles.

1. Anti-HIV drug discovery and development: current innovations and future trends;Zhan;J Med Chem,2016

2. The HIV therapy market;Gubernick;Nat Rev Drug Discovery,2016

3. Molecular basis of human immunodeficiency virus type 1 drug resistance: overview and recent developments;Menéndez-Arias;Antiviral Res,2013

4. Mechanistic study of common non-nucleoside reverse transcriptase inhibitor-resistant mutations with K103N and Y181C substitutions;Lai;Viruses,2016

5. Non-nucleoside reverse transcriptase inhibitors (NNRTIs), their discovery, development, and use in the treatment of HIV-1 infection: a review of the last 20 years (1989–2009);de Bethune;Antiviral Res,2010

Cited by 12 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Deciphering the enigmas of non‐nucleoside reverse transcriptase inhibitors (NNRTIs): A medicinal chemistry expedition towards combating HIV drug resistance;Medicinal Research Reviews;2024-08-26

2. Target-based drug design strategies to overcome resistance to antiviral agents: opportunities and challenges;Drug Resistance Updates;2024-03

3. Research Progress in HIV and Mycobacterium tuberculosis Inhibitors Containing Sulfonamide Moiety;Journal of Chemistry;2023-12-07

4. Strategies in the Design and Development of Non-Nucleoside Reverse Transcriptase Inhibitors (NNRTIs);Viruses;2023-09-25

5. Novel Sulfonamide Derivatives Containing a Piperidine Moiety as New Bactericide Leads for Managing Plant Bacterial Diseases;International Journal of Molecular Sciences;2023-03-20