Novel inhibitors of epidermal growth factor receptor: (4-(Arylamino)-7H-pyrrolo[2,3-d]pyrimidin-6-yl)(1H-indol-2-yl)methanones and (1H-indol-2-yl)(4-(phenylamino)thieno[2,3-d]pyrimidin-6-yl)methanones-Reference-Cited by-同舟云学术

Novel inhibitors of epidermal growth factor receptor: (4-(Arylamino)-7H-pyrrolo[2,3-d]pyrimidin-6-yl)(1H-indol-2-yl)methanones and (1H-indol-2-yl)(4-(phenylamino)thieno[2,3-d]pyrimidin-6-yl)methanones

Published:2012-01 Issue:1 Volume:20 Page:125-136
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Beckers Thomas,Sellmer Andreas,Eichhorn Emerich,Pongratz Herwig,Schächtele Christoph,Totzke Frank,Kelter Gerhard,Krumbach Rebekka,Fiebig Heinz-Herbert,Böhmer Frank-D.,Mahboobi Siavosh

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference22 articles.

1. Novel Bis(1H-indol-2-yl)methanones as Potent Inhibitors of FLT3 and Platelet-Derived Growth Factor Receptor Tyrosine Kinase

2. Epidermal growth factor receptor expression in breast cancer association with biologic phenotype and clinical outcomes

3. EGFR targeting drugs in the treatment of head and neck squamous cell carcinoma

4. EGFR(S) Inhibitors in the Treatment of Gastro-Intestinal Cancers: Whats New?

5. Targeting epidermal growth factor receptor: Central signaling kinase in lung cancer

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