Targeting the gatekeeper residue in phosphoinositide 3-kinases-Reference-Cited by-同舟云学术

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Targeting the gatekeeper residue in phosphoinositide 3-kinases

Published:2005-04 Issue:8 Volume:13 Page:2825-2836
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Alaimo Peter J.,Knight Zachary A.,Shokat Kevan M.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference40 articles.

1. Characterization of a conserved structural determinant controlling protein kinase sensitivity to selective inhibitors;Blencke;Chem. Biol.,2004

2. Structural basis for selective inhibition of Src family kinases by PP1;Liu;Chem. Biol.,1999

3. Therapeutic potential of phosphoinositide 3-kinase inhibitors;Ward;Chem. Biol.,2003

4. Isoform-specific phosphoinositide 3-kinase inhibitors as therapeutic agents;Ward;Curr. Opin. Pharmacol.,2003

5. Protein kinase inhibitors: insights into drug design from structure;Noble;Science,2004

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2. Data-oriented protein kinase drug discovery;European Journal of Medicinal Chemistry;2024-05

3. An unconventional gatekeeper mutation sensitizes inositol hexakisphosphate kinases to an allosteric inhibitor;eLife;2023-10-16

4. An unconventional gatekeeper mutation sensitizes inositol hexakisphosphate kinases to an allosteric inhibitor;eLife;2023-10-16

5. Structural pathway for class III PI 3-kinase activation by the myristoylated GTP-binding pseudokinase VPS15;2023-09-28

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