Synthesis and antitrypanosomal evaluation of derivatives of N-benzyl-1,2-dihydroquinolin-6-ols: Effect of core substitutions and salt formation-Reference-Cited by-同舟云学术

Synthesis and antitrypanosomal evaluation of derivatives of N-benzyl-1,2-dihydroquinolin-6-ols: Effect of core substitutions and salt formation

Published:2011-01 Issue:1 Volume:19 Page:513-523
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Reid Carolyn S.,Patrick Donald A.,He Shanshan,Fotie Jean,Premalatha Kokku,Tidwell Richard R.,Wang Michael Zhuo,Liu Qiang,Gershkovich Pavel,Wasan Kishor M.,Wenzler Tanja,Brun Reto,Werbovetz Karl A.

Funder

Bill and Melinda Gates Foundation

WHO/TDR

Neglected Global Diseases Initiative at the University of British Columbia

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference31 articles.

1. Treatment of human African trypanosomiasis—present situation and needs for research and development

2. Melarsoprol versus eflornithine for treating late-stage Gambian trypanosomiasis in the Republic of Congo

3. Nifurtimox-eflornithine combination therapy for second-stage African Trypanosoma brucei gambiense trypanosomiasis: a multicentre, randomised, phase III, non-inferiority trial

4. NECT trial: more than a small victory over sleeping sickness

5. New Treatment Option for Second-Stage African Sleeping Sickness: In Vitro and In Vivo Efficacy of Aza Analogs of DB289

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