Development of α-keto-based inhibitors of cruzain, a cysteine protease implicated in Chagas disease-Reference-Cited by-同舟云学术

Development of α-keto-based inhibitors of cruzain, a cysteine protease implicated in Chagas disease

Published:2005-03 Issue:6 Volume:13 Page:2141-2156
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Choe Youngchool,Brinen Linda S.,Price Mark S.,Engel Juan C.,Lange Meinolf,Grisostomi Corinna,Weston Scott G.,Pallai Peter V.,Cheng Hong,Hardy Larry W.,Hartsough David S.,McMakin Marsha,Tilton Robert F.,Baldino Carmen M.,Craik Charles S.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference40 articles.

1. World Health Organization: Special Program for Research and Training in Tropical Diseases (TDR)

2. Synthesis and Structure−Activity Relationship Study of Potent Trypanocidal Thio Semicarbazone Inhibitors of the Trypanosomal Cysteine Protease Cruzain

3. Cysteine protease inhibitors alter Golgi complex ultrastructure and function in Trypanosoma cruzi

4. Cysteine Protease Inhibitors Cure an Experimental Trypanosoma cruzi Infection

5. Proteolytic Activities in Cell Extracts ofTrypanosoma cruzi*

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