4-([1,2,4]Triazolo[1,5-a]pyridin-6-yl)-5(3)-(6-methylpyridin-2-yl)imidazole and -pyrazole derivatives as potent and selective inhibitors of transforming growth factor-β type I receptor kinase-Reference-Cited by-同舟云学术

4-([1,2,4]Triazolo[1,5-a]pyridin-6-yl)-5(3)-(6-methylpyridin-2-yl)imidazole and -pyrazole derivatives as potent and selective inhibitors of transforming growth factor-β type I receptor kinase

Published:2014-05 Issue:9 Volume:22 Page:2724-2732
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Jin Cheng Hua,Krishnaiah Maddeboina,Sreenu Domalapally,Subrahmanyam Vura Bala,Park Hyun-Ju,Park So-Jung,Sheen Yhun Yhong,Kim Dae-Kee

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference49 articles.

1. TGF-β signalling from cell membrane to nucleus through SMAD proteins

2. Smad-dependent and Smad-independent pathways in TGF-β family signalling

3. Transforming growth factor-beta and Smad signalling in kidney diseases. Review Article

4. Role of transforming growth factor-β in the progression of heart failure

5. Effect of TGF-?/Smad signaling pathway on lung myofibroblast differentiation

Cited by 34 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Synthesis and biological evaluation of sulfonamide derivatives containing imidazole moiety as ALK5 inhibitors;Molecular Diversity;2024-08-30

2. Advances in the discovery of activin receptor-like kinase 5 (ALK5) inhibitors;Bioorganic Chemistry;2024-06

3. Synthesis of amide derivatives containing the imidazole moiety and evaluation of their anti‐cardiac fibrosis activity;Archiv der Pharmazie;2024-04-28

4. Synthesis and anti-liver fibrosis activity of imidazole and thiazole compounds containing amino acids;European Journal of Medicinal Chemistry;2024-04

5. Design, Synthesis, and In Vitro Antiproliferative Activity of 4,5,6-Trisubstituted 2-Aminopyrimidines as Potential TGF-β Inhibitors;Russian Journal of Organic Chemistry;2024-04