Discovery of DB18, a potent inhibitor of CLK kinases with a high selectivity against DYRK1A kinase

Author:

Brahmaiah Dabbugoddu,Kanaka Durga Bhavani Anagani,Aparna Pasula,Sampath Kumar Nangunoori,Solhi Hélène,Le Guevel Rémy,Baratte Blandine,Ruchaud Sandrine,Bach Stéphane,Singh Jadav Surender,Raji Reddy Chada,Roisnel Thierry,Mosset Paul,Levoin Nicolas,Grée René

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference65 articles.

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2. (a) Ferguson FM, Gray NS, Kinase inhibitors: the road ahead. Nature Reviews Drug Discovery2018;17:353-377; (b) Laufer S, Briner K, Bajorath J, Georg GI, Wang S, New horizons in drug discovery–understanding and advancing kinase inhibitors. J. Med. Chem. 2020;63:7921-7922.

3. PKIDB: A curated, annotated and updated database of protein kinase inhibitors in clinical trials;Carles;Molecules,2018

4. Properties of FDA-approved small molecule protein kinase inhibitors;Roskoski;Pharmacol Res,2019

5. Targeting RNA splicing for disease therapy;Havens;Wiley Interdiscip Rev RNA,2013

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