Design, synthesis, and docking studies of quinazoline analogues bearing aryl semicarbazone scaffolds as potent EGFR inhibitors-Reference-Cited by-同舟云学术

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Design, synthesis, and docking studies of quinazoline analogues bearing aryl semicarbazone scaffolds as potent EGFR inhibitors

Published:2017-06 Issue:12 Volume:25 Page:3148-3157
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Tu Yuanbiao,Wang Caolin,Xu Shan,Lan Zhou,Li Wei,Han Jiaqian,Zhou Yuanzhang,Zheng Pengwu,Zhu Wufu

Funder

National Natural Science Funds

Natural Science Foundation of Jiangxi

Education Department of Jiangxi Province

Jiangxi Science & Technology Normal University

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference16 articles.

1. Dual targeting of HER1/EGFR and HER2 with cetuximab and trastuzumab in patients with metastatic pancreatic cancer after gemcitabine failure: results of the “THERAPY”phase 1-2 trial

2. Targeting EGFR/HER2 pathways enhances the antiproliferative effect of gemcitabine in biliary tract and gallbladder carcinomas

3. ERBB receptors and cancer: the complexity of targeted inhibitors

4. Reciprocal and Complementary Role of MET Amplification and EGFR T790M Mutation in Acquired Resistance to Kinase Inhibitors in Lung Cancer

5. A Chemical Tuned Strategy to Develop Novel Irreversible EGFR-TK Inhibitors with Improved Safety and Pharmacokinetic Profiles

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2. Design and synthesis of novel Thiazolo[5,4-b]pyridine derivatives as potent and selective EGFR-TK inhibitors targeting resistance Mutations in non-small cell lung cancer;European Journal of Medicinal Chemistry;2024-10

3. 6-Bromo quinazoline derivatives as cytotoxic agents: design, synthesis, molecular docking and MD simulation;BMC Chemistry;2024-07-04

4. QSAR Based Drug Repurposing: A New Paradigm in Breast Cancer Research;Indian Journal of Pharmaceutical Education and Research;2024-06-21

5. Discovery of new 2,4-diaminopyrimidines derivatives as EGFRT790M kinase inhibitors: a structure-based approach with DFT calculation, drug-likeness, ADME-toxicity properties evaluation and MD simulation;Journal of Umm Al-Qura University for Applied Sciences;2024-01-16

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