t -Butyl pyridine and phenyl C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists-Reference-Cited by-同舟云学术

t -Butyl pyridine and phenyl C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists

Published:2017-04 Issue:8 Volume:25 Page:2451-2462
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Lee Sunho,Kang Dong Wook,Ryu HyungChul,Kim Changhoon,Ann Jihyae,Lee Hobin,Kim Eunhye,Hong Sunhye,Choi Sun,Blumberg Peter M.,Frank-Foltyn Robert,Bahrenberg Gregor,Stockhausen Hannelore,Christoph Thomas,Lee Jeewoo

Funder

National Research Foundation

Ministry of Science, ICT and Future Planning

National Institutes of Health

Center for Cancer Research

National Cancer Institute

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference31 articles.

1. The Cloned Capsaicin Receptor Integrates Multiple Pain-Producing Stimuli

2. Vanilloid (Capsaicin) Receptors in Health and Disease

3. Structural insights into transient receptor potential vanilloid type 1 (TRPV1) from homology modeling, flexible docking, and mutational studies

4. Structure of the TRPV1 ion channel determined by electron cryo-microscopy

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