2-Oxoamide inhibitors of cytosolic group IVA phospholipase A2 with reduced lipophilicity-Reference-Cited by-同舟云学术

2-Oxoamide inhibitors of cytosolic group IVA phospholipase A2 with reduced lipophilicity

Published:2016-10 Issue:19 Volume:24 Page:4544-4554
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Antonopoulou Georgia,Magrioti Victoria,Kokotou Maroula G.,Nikolaou Aikaterini,Barbayianni Efrosini,Mouchlis Varnavas D.^ORCID,Dennis Edward A.,Kokotos George

Funder

European Union

Greek National Funds

NIH

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference40 articles.

1. Cytosolic phospholipase A2: physiological function and role in disease

2. Phospholipase A2 Enzymes: Physical Structure, Biological Function, Disease Implication, Chemical Inhibition, and Therapeutic Intervention

3. Phospholipase A2inhibitors as potential therapeutic agents for the treatment of inflammatory diseases

4. Phospholipase A2inhibitors for the treatment of inflammatory diseases: a patent review (2010 – present)

5. Slow- and tight-binding inhibitors of the 85-kDa human phospholipase A2

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