Discovery of 1,2,3,4-tetrahydropyrimido[1,2-a]benzimidazoles as novel class of corticotropin releasing factor 1 receptor antagonists-Reference-Cited by-同舟云学术

Discovery of 1,2,3,4-tetrahydropyrimido[1,2-a]benzimidazoles as novel class of corticotropin releasing factor 1 receptor antagonists

Published:2018-05 Issue:9 Volume:26 Page:2229-2250
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Kojima Takuto,Mochizuki Michiyo,Takai Takafumi^ORCID,Hoashi Yasutaka^ORCID,Morimoto Sachie,Seto Masaki,Nakamura Minoru,Kobayashi Katsumi,Sako Yuu,Tanaka Maiko,Kanzaki Naoyuki,Kosugi Yohei,Yano Takahiko,Aso Kazuyoshi

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference23 articles.

1. Characterization of a 41-residue ovine hypothalamic peptide that stimulates secretion of corticotropin and beta-endorphin;Vale;Science,1981

2. Physiology and pharmacology of corticotropin-releasing factor;Owen;Pharmacol Rev,1991

3. Recent advances in corticotropin-releasing factor receptor antagonists;Dzierba;Annu Rep Med Chem,2008

4. Corticotropin-releasing factor receptor antagonists;Gilligan;Expert Opin Ther Pat,2006

5. Corticotropin-releasing factor 1 receptor antagonists: a patent review;Williams;Expert Opin Ther Pat,2013

Cited by 21 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Visible Light-Induced Radical Cascade Difluoromethylation/Cyclization of Unactivated Alkenes: Access to CF₂H-Substituted Polycyclic Imidazoles;ACS Omega;2024-06-19

2. Synthesis of 3,4-dihydropyrimido[1,2-a]benzimidazoles, promising CRF1 receptor antagonists;Russian Chemical Bulletin;2024-04

3. Synthesis of benzimidazole-fused 1,4-benzoxazepines and benzosultams spiro-connected to a 2-oxindole core via a tandem epoxide-opening/S_NAr approach;Organic & Biomolecular Chemistry;2024

4. 2,4-Diaryl-pyrimido[1,2-a]benzimidazole derivatives as novel anticancer agents endowed with potent anti-leukemia activity: Synthesis, biological evaluation and kinase profiling;European Journal of Medicinal Chemistry;2023-10

5. Structure-based drug discovery of a corticotropin-releasing hormone receptor 1 antagonist using an X-ray free-electron laser;Experimental & Molecular Medicine;2023-09-01