Design and discovery of 5-hydroxy-6-oxo-1,6-dihydropyrimidine-4-carboxamide inhibitors of HIV-1 integrase

Author:

Zhang Daoguang,Debnath Bikash,Yu Shenghui,Sanchez Tino Wilson,Christ Frauke,Liu Yang,Debyser Zeger,Neamati Nouri,Zhao GuisenORCID

Funder

National Natural Science Foundation of China

NIH/NIAID

NIH F31

CHRP

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference43 articles.

1. Novel therapeutic strategies targeting HIV integrase

2. HIV-1 Integrase: Mechanism and Inhibitor Design;Neamati,2011

3. Molecular mechanisms in retrovirus DNA integration

4. HIV Integrase Inhibitors: From Diketoacids to Heterocyclic Templates: A History of HIV Integrase Medicinal Chemistry at Merck West Point and Merck Rome (IRBM) Leading to the Discovery of Raltegravir;Egbertson,2011

5. Discovery of Raltegravir, a Potent, Selective Orally Bioavailable HIV-Integrase Inhibitor for the Treatment of HIV-AIDS Infection

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