Discovery of BI 135585, an in vivo efficacious oxazinanone-based 11β hydroxysteroid dehydrogenase type 1 inhibitor-Reference-Cited by-同舟云学术

Discovery of BI 135585, an in vivo efficacious oxazinanone-based 11β hydroxysteroid dehydrogenase type 1 inhibitor

Published:2017-07 Issue:14 Volume:25 Page:3649-3657
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Zhuang Linghang,Tice Colin M.,Xu Zhenrong,Zhao Wei,Cacatian Salvacion,Ye Yuan-Jie,Singh Suresh B.,Lindblom Peter,McKeever Brian M.,Krosky Paula M.,Zhao Yi,Lala Deepak,Kruk Barbara A.,Meng Shi,Howard Lamont,Johnson Judith A.,Bukhtiyarov Yuri,Panemangalore Reshma,Guo Joan,Guo Rong,Himmelsbach Frank,Hamilton Bradford,Schuler-Metz Annette,Schauerte Heike,Gregg Richard,McGeehan Gerard M.,Leftheris Katerina,Claremon David A.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

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