Synthesis and biological evaluation of a series of flavone derivatives as potential radioligands for imaging the multidrug resistance-associated protein 1 (ABCC1/MRP1)-Reference-Cited by-同舟云学术

Synthesis and biological evaluation of a series of flavone derivatives as potential radioligands for imaging the multidrug resistance-associated protein 1 (ABCC1/MRP1)

Published:2006-03 Issue:5 Volume:14 Page:1599-1607
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Mavel Sylvie,Dikic Branko,Palakas Somchit,Emond Patrick,Greguric Ivan,de Gracia Adrienne Gomez,Mattner Filomena,Garrigos Manuel,Guilloteau Denis,Katsifis Andrew

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference25 articles.

1. The mdrl gene, responsible for multidrug-resistance, codes for P-glycoprotein

2. Overexpression of a transporter gene in a multidrug-resistant human lung cancer cell line

3. Flavonoids: A class of modulators with bifunctional interactions at vicinal ATP- and steroid-binding sites on mouse P-glycoprotein

4. Correlation between the Affinity of Flavonoids Binding to the Cytosolic Site of Leishmania tropica Multidrug Transporter and Their Efficiency To Revert Parasite Resistance to Daunomycin

5. Recent advances in the discovery of flavonoids and analogs with high-affinity binding to P-glycoprotein responsible for cancer cell multidrug resistance

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