Cell-based and in-silico studies on the high intrinsic activity of two boron-containing salbutamol derivatives at the human β2-adrenoceptor-Reference-Cited by-同舟云学术

Cell-based and in-silico studies on the high intrinsic activity of two boron-containing salbutamol derivatives at the human β2-adrenoceptor

Published:2012-01 Issue:2 Volume:20 Page:933-941
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Soriano-Ursúa Marvin A.,McNaught-Flores Daniel A.,Nieto-Alamilla Gustavo,Segura-Cabrera Aldo,Correa-Basurto José,Arias-Montaño José A.,Trujillo-Ferrara José G.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference54 articles.

1. β2-adrenoceptor agonists: current and future direction

2. Long-acting beta-agonists in the management of chronic obstructive pulmonary disease: current and future agents

3. The selectivity of β -adrenoceptor antagonists at the human β 1, β 2 and β 3 adrenoceptors

4. Synthesis, pharmacological and in silico evaluation of 1-(4-di-hydroxy-3,5-dioxa-4-borabicyclo[4.4.0]deca-7,9,11-trien-9-yl)-2-(tert-butylamino)ethanol, a compound designed to act as a β2 adrenoceptor agonist

5. Design, synthesis and in vitro evaluation of (R)-4-(2-(tert-butylamino)-1-hydroxyethyl)-2-(hydroxymethyl)phenyl hydrogen phenylboronate: A novel salbutamol derivative with high intrinsic efficacy on the β2 adrenoceptor

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