6-Hydrophobic aromatic substituent pyrimethamine analogues as potential antimalarials for pyrimethamine-resistant Plasmodium falciparum-Reference-Cited by-同舟云学术

6-Hydrophobic aromatic substituent pyrimethamine analogues as potential antimalarials for pyrimethamine-resistant Plasmodium falciparum

Published:2019-12 Issue:24 Volume:27 Page:115158
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Saepua Siriporn,Sadorn Karoon,Vanichtanankul Jarunee,Anukunwithaya Tosapol,Rattanajak Roonglawan,Vitsupakorn Danoo,Kamchonwongpaisan Sumalee,Yuthavong Yongyuth,Thongpanchang Chawanee

Funder

BIOTEC

NSTDA’s Cluster and Program Management

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference29 articles.

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3. A broad analysis of resistance development in the malaria parasite;Corey;Nat Commun.,2016

4. Amino acid changes linked to pyrimethamine resistance in the dihydrofolate reductase-thymidylate synthase gene of Plasmodium falciparum;Cowman;Proc Natl Acad Sci USA,1988

5. Mechanisms of resistance of Plasmodium falciparum to antimalarial drugs;Hyde;Microb Inf,2002

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