Preparation and biological evaluation of conformationally constrained BACE1 inhibitors-Reference-Cited by-同舟云学术

Preparation and biological evaluation of conformationally constrained BACE1 inhibitors

Published:2015-07 Issue:13 Volume:23 Page:3260-3268
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Winneroski Leonard L.,Schiffler Matthew A.,Erickson Jon A.,May Patrick C.,Monk Scott A.,Timm David E.,Audia James E.,Beck James P.,Boggs Leonard N.,Borders Anthony R.,Boyer Robert D.,Brier Richard A.,Hudziak Kevin J.,Klimkowski Valentine J.,Garcia Losada Pablo,Mathes Brian M.,Stout Stephanie L.,Watson Brian M.,Mergott Dustin J.

Funder

U.S. DOE

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference18 articles.

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3. Biochemistry of Amyloid -Protein and Amyloid Deposits in Alzheimer Disease

4. The secretases: enzymes with therapeutic potential in Alzheimer disease

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