Identification of trans-4-[1-[[7-fluoro-2-(1-methyl-3-indolyl)-6-benzoxazolyl]acetyl]-(4S)-fluoro-(2S)-pyrrolidinylmethoxy]cyclohexanecarboxylic acid as a potent, orally active VLA-4 antagonist-Reference-Cited by-同舟云学术

Identification of trans-4-[1-[[7-fluoro-2-(1-methyl-3-indolyl)-6-benzoxazolyl]acetyl]-(4S)-fluoro-(2S)-pyrrolidinylmethoxy]cyclohexanecarboxylic acid as a potent, orally active VLA-4 antagonist

Published:2012-02 Issue:3 Volume:20 Page:1201-1212
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Setoguchi Masaki,Iimura Shin,Sugimoto Yuuichi,Yoneda Yoshiyuki,Chiba Jun,Watanabe Toshiyuki,Muro Fumihito,Iigo Yutaka,Takayama Gensuke,Yokoyama Mika,Taira Tomoe,Aonuma Misato,Takashi Tohru,Nakayama Atsushi,Machinaga Nobuo

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference41 articles.

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