Aminopyrazolo[1,5-a]pyrimidines as potential inhibitors of Mycobacterium tuberculosis: Structure activity relationships and ADME characterization-Reference-Cited by-同舟云学术

Aminopyrazolo[1,5-a]pyrimidines as potential inhibitors of Mycobacterium tuberculosis: Structure activity relationships and ADME characterization

Published:2015-11 Issue:22 Volume:23 Page:7240-7250
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Soares de Melo Candice,Feng Tzu-Shean,van der Westhuyzen Renier,Gessner Richard K.,Street Leslie J.,Morgans Garreth L.,Warner Digby F.,Moosa Atica,Naran Krupa,Lawrence Nina,Boshoff Helena I.M.,Barry Clifton E.,Harris C. John,Gordon Richard,Chibale Kelly

Funder

Intramural Research Program of NIAID

Foundation for the National Institutes of Health

Bill & Melinda Gates Foundation

South African Medical Research Council (MRC)

South African Tuberculosis Research and Innovation Initiative (SATRII)

Strategic Health Innovation Partnerships (SHIP) initiative

The University of Cape Town

South African Medical Research Council

South African Research Chairs Initiative of the Department of Science and Technology

South African National Research Foundation

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference49 articles.

1. World Health Organization. Global Tuberculosis Report; Technical Report from the World Health Organization: Geneva, Switzerland, 2014; Available at http://www.who.int/tb/publications/global_report/en/index.html.

2. Tuberculosis: What We Don’t Know Can, and Does, Hurt Us

3. Viewpoint: Scientific dogmas, paradoxes and mysteries of latent Mycobacterium tuberculosis infection

4. Current Status and Research Strategies in Tuberculosis Drug Development

5. Treatment of tuberculosis: update 2010

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