Design, synthesis, and biological evaluation of novel 7-azaindolyl-heteroaryl-maleimides as potent and selective glycogen synthase kinase-3β (GSK-3β) inhibitors-Reference-Cited by-同舟云学术

Design, synthesis, and biological evaluation of novel 7-azaindolyl-heteroaryl-maleimides as potent and selective glycogen synthase kinase-3β (GSK-3β) inhibitors

Published:2004-06 Issue:12 Volume:12 Page:3167-3185
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

O'Neill David J.,Shen Lan,Prouty Catherine,Conway Bruce R.,Westover Lori,Xu Jun Z.,Zhang Han-Cheng,Maryanoff Bruce E.,Murray William V.,Demarest Keith T.,Kuo Gee-Hong

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference47 articles.

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3. Molecular cloning and expression of glycogen synthase kinase-3/factor A.

4. The multifaceted roles of glycogen synthase kinase 3β in cellular signaling

5. Glycogen synthase kinase 3: an emerging therapeutic target

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