Design, synthesis, and biological activity of substituted 2-amino-5-oxo-5H-chromeno[2,3-b]pyridine-3-carboxylic acid derivatives as inhibitors of the inflammatory kinases TBK1 and IKKε for the treatment of obesity-Reference-Cited by-同舟云学术

Design, synthesis, and biological activity of substituted 2-amino-5-oxo-5H-chromeno[2,3-b]pyridine-3-carboxylic acid derivatives as inhibitors of the inflammatory kinases TBK1 and IKKε for the treatment of obesity

Published:2018-11 Issue:20 Volume:26 Page:5443-5461
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Beyett Tyler S.,Gan Xinmin,Reilly Shannon M.,Gomez Andrew V.,Chang Louise,Tesmer John J.G.,Saltiel Alan R.,Showalter Hollis D.

Funder

National Institutes of Health

Michigan Economic Development Corporation

Michigan Technology Tri-Corridor

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

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