Methylation of imidazoline related compounds leads to loss of α2-adrenoceptor affinity. Synthesis and biological evaluation of selective I1 imidazoline receptor ligands-Reference-Cited by-同舟云学术

Methylation of imidazoline related compounds leads to loss of α2-adrenoceptor affinity. Synthesis and biological evaluation of selective I1 imidazoline receptor ligands

Published:2012-08 Issue:15 Volume:20 Page:4710-4715
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Schann Stephan,Greney Hugues,Gasparik Vincent,Dontenwill Monique,Rascente Carla,Lacroix Gabriel,Monassier Laurent,Bruban Véronique,Feldman Josiane,Ehrhardt Jean-Daniel,Bousquet Pascal

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

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5. Imidazoleacetic acid-ribotide: An endogenous ligand that stimulates imidazol(in)e receptors

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