Development of α1,6-fucosyltransferase inhibitors through the diversity-oriented syntheses of GDP-fucose mimics using the coupling between alkyne and sulfonyl azide-Reference-Cited by-同舟云学术

Development of α1,6-fucosyltransferase inhibitors through the diversity-oriented syntheses of GDP-fucose mimics using the coupling between alkyne and sulfonyl azide

Published:2017-06 Issue:11 Volume:25 Page:2844-2850
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Manabe Yoshiyuki,Kasahara Satomi,Takakura Yohei,Yang Xiaoxiao,Takamatsu Shinji,Kamada Yoshihiro,Miyoshi Eiji,Yoshidome Daisuke,Fukase Koichi

Funder

JSPS

Nagase Research Grant

Naito Research Grant

Nikki Saneyoshi Research Grant

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference58 articles.

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4. Fucose: biosynthesis and biological function in mammals

5. The α1-6-fucosyltransferase gene and its biological significance

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