Design, syntheses, and pharmacological characterization of 17-cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6α-(isoquinoline-3′-carboxamido)morphinan analogues as opioid receptor ligands-Reference-Cited by-同舟云学术

Design, syntheses, and pharmacological characterization of 17-cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6α-(isoquinoline-3′-carboxamido)morphinan analogues as opioid receptor ligands

Published:2015-04 Issue:8 Volume:23 Page:1701-1715
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Yuan Yunyun,Zaidi Saheem A.,Stevens David L.,Scoggins Krista L.,Mosier Philip D.,Kellogg Glen E.,Dewey William L.,Selley Dana E.,Zhang Yan

Funder

NIH/NIDA

NIH

National Center for Research Resources Award

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference67 articles.

1. Expression of the μ-Opioid Receptor in CHO Cells: Ability of μ-Opioid Ligands to Promote α-Azidoanilido[32P]GTP Labeling of Multiple G Protein α Subunits

2. Single potassium channels opened by opioids in rat locus ceruleus neurons.

3. µ-Opioid Receptor Modulates Peptide Release From Rat Neurohypophysial Terminals By Inhibiting Ca2+ Influx

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