Modulation of opioid receptor affinity and efficacy via N-substitution of 9β-hydroxy-5-(3-hydroxyphenyl)morphan: Synthesis and computer simulation study-Reference-Cited by-同舟云学术

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Modulation of opioid receptor affinity and efficacy via N-substitution of 9β-hydroxy-5-(3-hydroxyphenyl)morphan: Synthesis and computer simulation study

Published:2017-04 Issue:8 Volume:25 Page:2406-2422
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Truong Phong M.,Hassan Sergio A.,Lee Yong-Sok,Kopajtic Theresa A.,Katz Jonathan L.,Chadderdon Aaron M.,Traynor John R.,Deschamps Jeffrey R.,Jacobson Arthur E.,Rice Kenner C.

Funder

NIH

National Institute on Drug Abuse

National Institute of Alcohol Abuse and Alcoholism

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference35 articles.

1. Biased agonism: An emerging paradigm in GPCR drug discovery

2. Unravelling intrinsic efficacy and ligand bias at G protein coupled receptors: A practical guide to assessing functional data

3. Fulfilling the Promise of "Biased" G Protein–Coupled Receptor Agonism

4. Ligand-Based Discovery of a New Scaffold for Allosteric Modulation of the μ-Opioid Receptor

5. Biased Agonism of Endogenous Opioid Peptides at the μ-Opioid Receptor

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1. Alkoxy chain length governs the potency of 2-benzylbenzimidazole ‘nitazene’ opioids associated with human overdose;Psychopharmacology;2023-09-02

2. Morphine alkaloids: History, biology, and synthesis;The Alkaloids: Chemistry and Biology;2021

3. Pharmacodynamics and pharmacokinetics of the novel synthetic opioid, U-47700, in male rats;Neuropharmacology;2020-10

4. The Intriguing Effects of Substituents in the N-Phenethyl Moiety of Norhydromorphone: A Bifunctional Opioid from a Set of “Tail Wags Dog” Experiments;Molecules;2020-06-06

5. Endogenous opiates and behavior: 2017;Peptides;2020-02

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