Synthesis of a [6- Pyridinyl - 18 F]-labelled fluoro derivative of WAY-100635 as a candidate radioligand for brain 5-HT 1A receptor imaging with PET-Reference-Cited by-同舟云学术

Synthesis of a [6- Pyridinyl - 18 F]-labelled fluoro derivative of WAY-100635 as a candidate radioligand for brain 5-HT 1A receptor imaging with PET

Published:2003-07 Issue:13 Volume:11 Page:2769-2782
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Karramkam Mylène,Hinnen Françoise,Berrehouma Myriam,Hlavacek Christophe,Vaufrey Françoise,Halldin Christer,McCarron Julie A.,Pike Victor W.,Dollé Frédéric

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference61 articles.

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2. Neuroimaging of mood disorders

3. Brain Serotonin1A Receptor Binding Measured by Positron Emission Tomography With [11C]WAY-100635

4. Pindolol binding to 5-HT 1A receptors in the human brain confirmed with positron emission tomography

5. Pindolol Augmentation of Selective Serotonin Reuptake Inhibitors: PET Evidence That the Dose Used in Clinical Trials Is Too Low

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