Assessment of the combined approach of N-alkylation and salt formation to enhance aqueous solubility of tertiary amines using bupivacaine as a model drug
Author:
Publisher
Elsevier BV
Subject
Pharmaceutical Science
Reference39 articles.
1. Salt selection and optimization procedures for pharmaceutical new chemical entities;Bastin;Org. Process Res. Dev.,2000
2. Transdermal delivery of 5-fluorouracil (5-FU) through hairless mouse skin by 1-alkyloxycarbonyl-5-FU prodrugs: physicochemical characterization of prodrugs and correlations with transdermal delivery;Beall;Int. J. Pharm.,1994
3. Salt forms of drugs and absorption;Bighley,1995
4. Novel approaches in prodrug design;Bodor;Drugs Future,1981
5. Prodrugs of 5-fluorouracil V 1-Alkoxycarbonyl derivatives as potential prodrug forms for improved rectal or oral delivery of 5-fluorouracil;Buur;J. Pharm. Sci.,1986
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