Prediction of blood–brain barrier permeation of α-adrenergic and imidazoline receptor ligands using PAMPA technique and quantitative-structure permeability relationship analysis-Reference-Cited by-同舟云学术

Prediction of blood–brain barrier permeation of α-adrenergic and imidazoline receptor ligands using PAMPA technique and quantitative-structure permeability relationship analysis

Published:2015-02 Issue: Volume:68 Page:94-105
ISSN:0928-0987
Container-title:European Journal of Pharmaceutical Sciences
language:en
Short-container-title:European Journal of Pharmaceutical Sciences

Author:

Vucicevic Jelica,Nikolic Katarina,Dobričić Vladimir,Agbaba Danica

Funder

Ministry of Education, Science and Technological Development of the Republic of Serbia

Publisher

Elsevier BV

Subject

Pharmaceutical Science

Reference58 articles.

1. Prediction of blood–brain barrier permeation in drug discovery from in vivo, in vitro and in silico models;Abbott;Drug Discov. Today Technol.,2004

2. Astrocyte–endothelial interactions at the blood–brain barrier;Abbott;Nat. Rev. Neurosci.,2006

3. APPENDIX D. 2008. Descriptor (Optional)-Cadaster..

4. Absorption and Drug Development;Avdeef,2003

5. The rise of PAMPA;Avdeef;Expert Opin. Drug Metab. Toxicol.,2005

Cited by 28 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Design, synthesis and biological evaluation of N-salicyloyl tryptamine derivatives as multifunctional neuroprotectants for the treatment of ischemic stroke;European Journal of Medicinal Chemistry;2024-11

2. Modelling of chromatographic and electrophoretic behaviour of imidazoline and alpha adrenergic receptors ligands under different acid-base conditions;ADMET and DMPK;2024-05-04

3. First report on pesticide sub-chronic and chronic toxicities against dogs using QSAR and chemical read-across;SAR and QSAR in Environmental Research;2024-02-23

4. Design, Synthesis, In Silico Studies and In Vitro Evaluation of New Indole- and/or Donepezil-like Hybrids as Multitarget-Directed Agents for Alzheimer’s Disease;Pharmaceuticals;2023-08-22

5. In vitro and in silico computational methods for assessing vaginal permeability;Drug Development and Industrial Pharmacy;2023-03-04