Guggulsterone antagonizes farnesoid X receptor induction of bile salt export pump but activates pregnane X receptor to inhibit cholesterol 7α-hydroxylase gene
Author:
Publisher
Elsevier BV
Subject
Cell Biology,Molecular Biology,Biochemistry,Biophysics
Reference17 articles.
1. Bile acid regulation of gene expression: roles of nuclear hormone receptors;Chiang;Endocr. Rev.,2002
2. Bile acid regulation of hepatic physiology: III. Bile acids and nuclear receptors;Chiang;Am. J. Physiol. Gastrointest. Liver Physiol.,2003
3. A regulatory cascade of the nuclear receptors FXR, SHP-1, and LRH-1 represses bile acid biosynthesis;Goodwin;Mol. Cell,2000
4. Molecular basis for feedback regulation of bile acid synthesis by nuclear receptors;Lu;Mol. Cell,2000
5. Human bile salt export pump (BSEP) promoter is transactivated by the farnesoid X receptor/bile acid receptor (FXR/BAR);Ananthanarayanan;J. Biol. Chem.,2001
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