Characterisation of the binding of [3H]MDL 105,519, a radiolabelled antagonist for the N-methyl-d-aspartate-associated glycine site, to pig cortical brain membranes-Reference-Cited by-同舟云学术

Characterisation of the binding of [3H]MDL 105,519, a radiolabelled antagonist for the N-methyl-d-aspartate-associated glycine site, to pig cortical brain membranes

Published:1997-04 Issue:2 Volume:226 Page:79-82
ISSN:0304-3940
Container-title:Neuroscience Letters
language:en
Short-container-title:Neuroscience Letters

Author:

Höfner G,Wanner K.Th

Publisher

Elsevier BV

Subject

General Neuroscience

Reference19 articles.

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2. Baron, B.M., Siegel, B.W., Parrison, B.L., Kehne, J.H., McCloskey, T.C., Schmidt, C.J., Taylor, V.L., Fadayel, G.M., Murawski, M.K., van Giersbergen, P.L.M., White, H.S. and Salituro, F.G., Pharmacological characterisation of MDL105,519 a systemically active antagonist of the NMDA receptor-associated glycine recognition site, Soc. Neurosci. Abstr., 21 (1995) 436.9.

3. [3H]5,7-Dichlorokynurenic acid, a novel radioligand labels NMDA receptor-associated glycine binding sites;Baron;Eur. J. Pharmacol.,1991

4. Polyamine-directed non-competitive NMDA antagonists;Carter;Mol. Neuropharmacol.,1992

5. Relationship between the inhibition constant (Ki) and the concentration of inhibitor which causes 50 per cent inhibition (IC50) of an enzymatic reaction;Cheng;Biochem. Pharmacol.,1973

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