Benzoflavone activators of the cystic fibrosis transmembrane conductance regulator: towards a pharmacophore model for the nucleotide-binding domain

Author:

Springsteel Mark F,Galietta Luis J.V,Ma Tonghui,By Kolbot,Berger Gideon O,Yang Hong,Dicus Christopher W,Choung Wonken,Quan Chao,Shelat Anang A,Guy R.Kiplin,Verkman A.S,Kurth Mark J,Nantz Michael H

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference29 articles.

1. Young, L. Y.; Koda-Kimble, M. A. Applied Therapeutics, The Clinical Use of Drugs, 6th Ed.; Applied Theraputics: Vancouver, NA, 1995; p 100.1.

2. Role of CFTR in Airway Disease

3. An algorithm for finding protein–DNA binding sites with applications to chromatin- immunoprecipitation microarray experiments

4. Gene therapy for cystic fibrosis

5. FDA Halts All Gene Therapy Trials at Penn

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