Synthesis of N -substituted piperidine-4-(benzylidene-4-carboxylic acids) and evaluation as inhibitors of steroid-5α-reductase type 1 and 2-Reference-Cited by-同舟云学术

Synthesis of N -substituted piperidine-4-(benzylidene-4-carboxylic acids) and evaluation as inhibitors of steroid-5α-reductase type 1 and 2

Published:2000-06 Issue:6 Volume:8 Page:1479-1487
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Picard Franck,Baston Eckhard,Reichert Wolfgang,Hartmann Rolf W.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference30 articles.

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3. 5α-Reductase inhibitors in prostate cancer;Gormley;Endocrine-Related Cancer,1996

4. The effect of finasteride, a 5 alpha-reductase inhibitor, on scalp skin testosterone and dihydrotestosterone concentrations in patients with male pattern baldness;Dallob;J. Clin. Endocrinol. Metab.,1994

5. 5α-Reductase activity in idiopathic hirsutism;Serafini;Fertil. Steril.,1985

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