Human Muscarinic Receptor Binding Characteristics of Antimuscarinic Agents to Treat Overactive Bladder

Author:

Maruyama Shuji1,Oki Tomomi1,Otsuka Atsushi2,Shinbo Hitoshi2,Ozono Seiichiro2,Kageyama Shinji3,Mikami Yuuki4,Araki Isao4,Takeda Masayuki4,Masuyama Keisuke5,Yamada Shizuo1

Affiliation:

1. Department of Pharmacokinetics and Pharmacodynamics and COE Program in the 21st Century, School of Pharmaceutical Sciences, University of Shizuoka, Shizuoka

2. Department of Urology, Hamamatsu University School of Medicine, Hamamatsu

3. Shio Urologic Clinic, Shizuoka, University of Yamanashi, Tamaho, Japan

4. Department of Urology, School of Medicine, University of Yamanashi, Tamaho, Japan

5. Department of Orolaryngology, School of Medicine, University of Yamanashi, Tamaho, Japan

Publisher

Ovid Technologies (Wolters Kluwer Health)

Subject

Urology

Reference20 articles.

1. International Union of Pharmacology. XVII. Classification of muscarinic acetylcholine receptors;Caulfield;Pharmacol Rev,1998

2. Differential gene expression of cholinergic muscarinic receptor subtypes in male and female normal human urinary bladder;Sigala;Urology,2002

3. Pharmacology of lower urinary tract smooth muscles and penile erectile tissues;Andersson;Pharmacol Rev,1993

4. Muscarinic acetylcholine receptor subtypes mediating urinary bladder contractility and coupling to GTP binding proteins;Wang;J Pharmacol Exp Ther,1995

5. A placebo-controlled, multicentre study comparing the tolerability and efficacy of propiverine and oxybutynin in patients with urgency and urge incontinence;Madersbacher;BJU Int,1999

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