Assessment of Inverse Agonism for the Angiotensin II Type 1 Receptor
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Elsevier
Reference22 articles.
1. The conformational change responsible for AT1 receptor activation is dependent upon two juxtaposed asparagine residues on transmembrane helices III and VII;Balmforth;J. Biol. Chem.,1997
2. Recent developments in constitutive receptor activity and inverse agonism, and their potential for GPCR drug discovery;Bond;Trends Pharmacol. Sci.,2006
3. Constitutive activation of the angiotensin II type 1 receptor alters the spatial proximity of transmembrane 7 to the ligand-binding pocket;Boucard;J. Biol. Chem.,2003
4. Mechanism of constitutive activation of the AT1 receptor: Influence of the size of the agonist switch binding residue Asn(111);Feng;Biochemistry,1998
5. Mutation of Asn111 in the third transmembrane domain of the AT1A angiotensin II receptor induces its constitutive activation;Groblewski;J. Biol. Chem.,1997
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