Development and profiling of mGlu7 NAMs with a range of saturable inhibition of agonist responses in vitro-Reference-Cited by-同舟云学术

Development and profiling of mGlu7 NAMs with a range of saturable inhibition of agonist responses in vitro

Published:2022-10 Issue: Volume:74 Page:128923
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Reed Carson W.,Rodriguez Alice L.,Kalbfleisch Jacob J.,Seto Mabel,Jenkins Matthew T.,Blobaum Anna L.,Chang Sichen,Lindsley Craig W.,Niswender Colleen M.

Funder

National Institute of Mental Health

Congressionally Directed Medical Research Programs

National Institutes of Health

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference25 articles.

1. Metabotropic Glutamate Receptors: Physiology, Pharmacology, and Disease

2. Constitutive activity of metabotropic glutamate receptor 7

3. Phasic and Tonic mGlu7 Receptor Activity Modulates the Thalamocortical Network

4. Enrichment of mGluR7a in the Presynaptic Active Zones of GABAergic and Non-GABAergic Terminals on Interneurons in the Rat Somatosensory Cortex

5. High level of mGluR7 in the presynaptic active zones of select populations of GABAergic terminals innervating interneurons in the rat hippocampus

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1. dx.doi.org/10.1124/molpharm.123.000678Pharmacol104:17-27, July 2023;MOL PHARMACOL;2023

2. Differential Activity of Orthosteric Agonists and Allosteric Modulators at Metabotropic Glutamate Receptor 7;Molecular Pharmacology;2023-04-27

3. Differential activity of mGlu7 allosteric modulators provides evidence for mGlu7/8 heterodimers at hippocampal Schaffer collateral-CA1 synapses;Journal of Biological Chemistry;2022-10