Discovery of novel benzylidene-1,3-thiazolidine-2,4-diones as potent and selective inhibitors of the PIM-1, PIM-2, and PIM-3 protein kinases-Reference-Cited by-同舟云学术

Discovery of novel benzylidene-1,3-thiazolidine-2,4-diones as potent and selective inhibitors of the PIM-1, PIM-2, and PIM-3 protein kinases

Published:2012-07 Issue:14 Volume:22 Page:4599-4604
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Dakin Les A.,Block Michael H.,Chen Huawei,Code Erin,Dowling James E.,Feng Xiaomei,Ferguson Andrew D.,Green Isabelle,Hird Alexander W.,Howard Tina,Keeton Erika K.,Lamb Michelle L.,Lyne Paul D.,Pollard Hannah,Read Jon,Wu Allan J.,Zhang Tao,Zheng Xiaolan

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference32 articles.

1. Murine leukemia virus-induced T-cell lymphomagenesis: Integration of proviruses in a distinct chromosomal region

2. Predisposition to lymphomagenesis in pim-1 transgenic mice: Cooperation with c-myc and N-myc in murine leukemia virus-induced tumors

3. Pim-1: A serine/threonine kinase with a role in cell survival, proliferation, differentiation and tumorigenesis

4. Structural Basis of Constitutive Activity and a Unique Nucleotide Binding Mode of Human Pim-1 Kinase

5. For better or for worse: the role of Pim oncogenes in tumorigenesis

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