Discovery and structure–activity relationships of pentanedioic acid diamides as potent inhibitors of 11β-hydroxysteroid dehydrogenase type I-Reference-Cited by-同舟云学术

Discovery and structure–activity relationships of pentanedioic acid diamides as potent inhibitors of 11β-hydroxysteroid dehydrogenase type I

Published:2009-05 Issue:10 Volume:19 Page:2674-2678
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Roche Didier,Carniato Denis,Leriche Caroline,Lepifre Franck,Christmann-Franck Serge,Graedler Ulrich,Charon Christine,Bozec Sophie,Doare Liliane,Schmidlin Fabien,Lecomte Marc,Valeur Eric

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference44 articles.

1. Metabolic conversion as a pre-receptor control mechanism for lipophilic hormones

2. 11β-Hydroxysteroid Dehydrogenase Type 1: A Tissue-Specific Regulator of Glucocorticoid Response

3. Hypertension in mice lacking 11β-hydroxysteroid dehydrogenase type 2

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