Identification of 9-fluoro substituted (−)-cytisine derivatives as ligands with high affinity for nicotinic receptors-Reference-Cited by-同舟云学术

Identification of 9-fluoro substituted (−)-cytisine derivatives as ligands with high affinity for nicotinic receptors

Published:2010-11 Issue:22 Volume:20 Page:6667-6670
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Houllier Nicolas,Gopisetti JaganMohan,Lestage Pierre,Lasne Marie-Claire,Rouden Jacques

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference42 articles.

1. O’Neill, B. T. Pyridone-Fused Azabicyclic- or Cytisine derivatives, their Preparation and their Use in Addiction Therapy. (a) PCT Int. Appl. 1998, WO9818,798,1998; Chem. Abstr. 1998, 119, 4774k. (b) U.S. Patent 6,235,734B1, 2001.

2. Synthesis and preliminary pharmacological evaluation of some cytisine derivatives

3. Synthesis of Analogues of (−)-Cytisine for in Vivo Studies of Nicotinic Receptors Using Positron Emission Tomography

4. Nicotinic receptor binding of [3H]cytisine, [3H]nicotine and [3H]methylcarbamylcholine in rat brain

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