Discovery of an l-alanine ester prodrug of the Hsp90 inhibitor, MPC-3100-Reference-Cited by-同舟云学术

Discovery of an l-alanine ester prodrug of the Hsp90 inhibitor, MPC-3100

Published:2015-11 Issue:22 Volume:25 Page:5254-5257
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Kim Se-Ho,Tangallapally Rajendra,Kim In Chul,Trovato Richard,Parker Daniel,Patton J. Scott,Reeves Leslie,Bradford Chad,Wettstein Daniel,Baichwal Vijay,Papac Damon,Bajji Ashok,Carlson Robert,Yager Kraig M.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference19 articles.

1. New Paradigms in Anticancer Therapy: Targeting Multiple Signaling Pathways With Kinase Inhibitors

2. Targeting cell signaling pathways for drug discovery: An old lock needs a new key

3. Drug resistance in cancer: Principles of emergence and prevention

4. Hsp90, an unlikely ally in the war on cancer

5. HSP90 inhibition: two-pronged exploitation of cancer dependencies

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