TR-FRET binding assay targeting unactivated form of Bruton’s tyrosine kinase
Author:
Publisher
Elsevier BV
Subject
Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry
Reference14 articles.
1. The tyrosine kinase network regulating mast cell activation
2. Targeting Bruton's tyrosine kinase in B cell malignancies
3. Tec Family Kinases in Inflammation and Disease
4. Measuring and interpreting the selectivity of protein kinase inhibitors
5. Rational design of inhibitors that bind to inactive kinase conformations
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1. Screening assays for tyrosine kinase inhibitors: A review;Journal of Pharmaceutical and Biomedical Analysis;2023-01
2. Discovery of a potent BTK and IKZF1/3 triple degrader through reversible covalent BTK PROTAC development;Current Research in Chemical Biology;2022
3. Compound Screening;Reference Module in Biomedical Sciences;2021
4. Design and Synthesis of Novel Amino-triazine Analogues as Selective Bruton’s Tyrosine Kinase Inhibitors for Treatment of Rheumatoid Arthritis;Journal of Medicinal Chemistry;2018-09-14
5. Design and synthesis of novel pyrimidine analogs as highly selective, non-covalent BTK inhibitors;Bioorganic & Medicinal Chemistry Letters;2018-01
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