7-Azaindole-3-acetic acid derivatives: Potent and selective CRTh2 receptor antagonists-Reference-Cited by-同舟云学术

7-Azaindole-3-acetic acid derivatives: Potent and selective CRTh2 receptor antagonists

Published:2009-08 Issue:16 Volume:19 Page:4794-4798
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Sandham David A.,Adcock Claire,Bala Kamlesh,Barker Lucy,Brown Zarin,Dubois Gerald,Budd David,Cox Brian,Fairhurst Robin A.,Furegati Markus,Leblanc Catherine,Manini Jodie,Profit Rachael,Reilly John,Stringer Rowan,Schmidt Alfred,Turner Katharine L.,Watson Simon J.,Willis Jennifer,Williams Gareth,Wilson Caroline

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference25 articles.

1. Release of Prostaglandin D2into Human Airways during Acute Antigen Challenge

2. Antagonism of the prostaglandin D2 receptors DP1 and CRTH2 as an approach to treat allergic diseases

3. A small molecule CRTH2 antagonist inhibits FITC-induced allergic cutaneous inflammation

4. An Orally Bioavailable Small Molecule Antagonist of CRTH2, Ramatroban (BAY u3405), Inhibits Prostaglandin D2-Induced Eosinophil Migration in Vitro

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