Synthesis and preclinical evaluation of [18F]FSL25.1188, a reversible PET radioligand for monoamine oxidase-B-Reference-Cited by-同舟云学术

Synthesis and preclinical evaluation of [18F]FSL25.1188, a reversible PET radioligand for monoamine oxidase-B

Published:2019-07 Issue:13 Volume:29 Page:1624-1627
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Dahl Kenneth,Bernard-Gauthier Vadim,Nag Sangram,Varnäs Katarina,Narayanaswami Vidya,Mahdi Moein Mohammad,Arakawa Ryosuke,Vasdev Neil^ORCID,Halldin Christer

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference23 articles.

1. Localization of monoamine oxidases in human peripheral tissues

2. Distinct monoamine oxidase A and B populations in primate brain

3. Increased monoamine oxidase b activity in plaque-associated astrocytes of Alzheimer brains revealed by quantitative enzyme radioautography

4. Evidence for Astrocytosis in Prodromal Alzheimer Disease Provided by 11C-Deuterium-L-Deprenyl: A Multitracer PET Paradigm Combining 11C-Pittsburgh Compound B and 18F-FDG

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