Design, synthesis and biological evaluation of a bivalent μ opiate and adenosine A1 receptor antagonist-Reference-Cited by-同舟云学术

Design, synthesis and biological evaluation of a bivalent μ opiate and adenosine A1 receptor antagonist

Published:2009-12 Issue:23 Volume:19 Page:6736-6739
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Mathew Smitha C.,Ghosh Nandita,By Youlet,Berthault Aurélie,Virolleaud Marie-Alice,Carrega Louis,Chouraqui Gaëlle,Commeiras Laurent,Condo Jocelyne,Attolini Mireille,Gaudel-Siri Anouk,Ruf Jean,Parrain Jean-Luc,Rodriguez Jean,Guieu Régis

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference28 articles.

1. Opioid agonist and antagonist bivalent ligands. The relationship between spacer length and selectivity at multiple opioid receptors

2. A Novel Pharmacological Approach to Treating Cardiac Ischemia

3. A Bivalent Ligand (KDAN-18) Containing δ-Antagonist and κ-Agonist Pharmacophores Bridges δ2 and κ1 Opioid Receptor Phenotypes

4. Novel and potent tacrine-related hetero- and homobivalent ligands for acetylcholinesterase and butyrylcholinesterase

5. Synthesis and Preliminary In vitro Investigation of Bivalent Ligands Containing Homo- and Heterodimeric Pharmacophores at μ, δ, and κ Opioid Receptors

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