Trifluoromethyl group as a pharmacophore: Effect of replacing a CF3 group on binding and agonist activity of a glucocorticoid receptor ligand-Reference-Cited by-同舟云学术

Trifluoromethyl group as a pharmacophore: Effect of replacing a CF3 group on binding and agonist activity of a glucocorticoid receptor ligand

Published:2005-11 Issue:21 Volume:15 Page:4761-4769
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Betageri Raj,Zhang Yan,Zindell Renee M.,Kuzmich Daniel,Kirrane Thomas M.,Bentzien Jörg,Cardozo Mario,Capolino Alison J.,Fadra Tazmeen N.,Nelson Richard M.,Paw Zofia,Shih Daw-Tsun,Shih Cheng-Kon,Zuvela-Jelaska Ljiljana,Nabozny Gerald,Thomson David S.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference44 articles.

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4. Glucocorticoids;Toogood,2001

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