Design and synthesis of AX4697, a bisindolylmaleimide exo-affinity probe that labels protein kinase C alpha and beta-Reference-Cited by-同舟云学术

Design and synthesis of AX4697, a bisindolylmaleimide exo-affinity probe that labels protein kinase C alpha and beta

Published:2008-11 Issue:22 Volume:18 Page:5955-5958
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Liu Yongsheng,Wu Jiangyue,Weissig Helge,Betancort Juan M.,Gai Wen Zhi,Leventhal Phillip S.,Patricelli Matthew P.,Samii Babak,Szardenings Anna K.,Shreder Kevin R.,Kozarich John W.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference25 articles.

1. Functional Interrogation of the Kinome Using Nucleotide Acyl Phosphates

2. Wortmannin, a Widely Used Phosphoinositide 3-Kinase Inhibitor, also Potently Inhibits Mammalian Polo-like Kinase

3. A Cell-permeable, Activity-based Probe for Protein and Lipid Kinases

4. Synthesis of AX7593, a Quinazoline-Derived Photoaffinity Probe for EGFR

5. Structure-guided development of affinity probes for tyrosine kinases using chemical genetics

Cited by 5 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Design, synthesis, and evaluation of cell permeable probes for protein kinases;Tetrahedron;2016-01

2. Detection of ubiquitin–proteasome enzymatic activities in cells: Application of activity-based probes to inhibitor development;Biochimica et Biophysica Acta (BBA) - Molecular Cell Research;2012-11

3. A Peptide Photoaffinity Probe Specific for the Active Conformation of the Abl Tyrosine Kinase;ChemBioChem;2012-10-18

4. Irreversible Protein Kinase Inhibitors: Balancing the Benefits and Risks;Journal of Medicinal Chemistry;2012-06-08

5. New indole amide derivatives as potent CRTH2 receptor antagonists;Bioorganic & Medicinal Chemistry Letters;2011-06