In vitro and in silico PTP-1B inhibition and in vivo antidiabetic activity of semisynthetic moronic acid derivatives

Author:

Cerón-Romero Litzia,Paoli PaoloORCID,Camici GuidoORCID,Flores-Morales Virginia,Rios María Yolanda,Ramírez-Espinosa Juan J.,Hidalgo-Figueroa Sergio,Navarrete-Vázquez Gabriel,Estrada-Soto SamuelORCID

Funder

Facultad de Farmacia

SEP-CONACyT Ciencia Básica

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference17 articles.

1. Discovery of Thiazolidine-2,4-Dione/Biphenylcarbonitrile Hybrid as Dual PPAR α/γ Modulator with Antidiabetic Effect:In vitro, In SilicoandIn VivoApproaches

2. WHO Fact sheet #312 January 2015 [on line September 28th 2014, http://www.who.int/mediacentre/factsheets/fs312/en/].

3. ADA Diabetes care volume 37, supplement 1, January 2014 [on line October 28th 2014, http://care.diabetesjournals.org/content/37/Supplement_1/S14.extract].

4. IDF Atlas Sixth edition 2013 [on line September 22th 2014 www.idf.org/diabetesatlas].

5. Recent Advances in Therapeutic Approaches toType 2 Diabetes

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