4-Phenyl-1,2,3,6-tetrahydropyridine, an excellent fragment to improve the potency of PARP-1 inhibitors-Reference-Cited by-同舟云学术

4-Phenyl-1,2,3,6-tetrahydropyridine, an excellent fragment to improve the potency of PARP-1 inhibitors

Published:2005-10 Issue:19 Volume:15 Page:4221-4225
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Ishida Junya,Hattori Kouji,Yamamoto Hirofumi,Iwashita Akinori,Mihara Kayoko,Matsuoka Nobuya

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference24 articles.

1. Pharmacological Modulation of Poly(ADP-ribose) Polymerase-Mediated Cell Death: Exploitation in Cancer Chemotherapy

2. Chiarugi, I. TIPS 2002, 23, 122; Szabó, C.; Virag, L. Pharmacol. Rev. 2002, 54, 375.

3. de Murcia, G., Shall, S. Eds; From DNA Damage and Stress Signaling to Cell Death: Poly ADP-ribosylation Reactions; Oxford University Press: Oxford, 2000.

4. Szabó, C., Ed.; Cell Death: The Role of PARP; CRC Press: Boca Raton, FL, 2000 and references therein.

5. Activation of Poly(ADP-Ribose) Polymerase in the Rat Hippocampus May Contribute to Cellular Recovery Following Sublethal Transient Global Ischemia

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