Pyrimido[4,5-d]azepines as potent and selective 5-HT2C receptor agonists: Design, synthesis, and evaluation of PF-3246799 as a treatment for urinary incontinence-Reference-Cited by-同舟云学术

Pyrimido[4,5-d]azepines as potent and selective 5-HT2C receptor agonists: Design, synthesis, and evaluation of PF-3246799 as a treatment for urinary incontinence

Published:2011-05 Issue:9 Volume:21 Page:2715-2720
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Andrews Mark D.,Fish Paul V.,Blagg Julian,Brabham Tiffini K.,Brennan Paul E.,Bridgeland Alison,Brown Alan D.,Bungay Peter J.,Conlon Kelly M.,Edmunds Nicholas J.,af Forselles Kerry,Gibbons Colleen P.,Green Martin P.,Hanton Giles,Holbrook Mark,Jessiman Alan S.,McIntosh Karin,McMurray Gordon,Nichols Carly L.,Root James A.,Storer R. Ian,Sutton Michael R.,Ward Robin V.,Westbrook Dominique,Whitlock Gavin A.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference45 articles.

1. Anti-obesity pharmacotherapy: Future perspectives utilising 5-HT2C receptor agonists

2. The potential use of selective 5-HT2Cagonists in treating obesity

3. 5-HT2C receptor agonists as an innovative approach for psychiatric disorders

4. Investigation of the role of 5-HT2receptor subtypes in the control of the bladder and the urethra in the anaesthetized female rat

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