Steroidal C-21 heteroaryl thioethers. Part 3: Pregn-4-eno-[3,2-c]pyrazole fused A ring modified steroids as selective glucocorticoid receptor modulators (dissociated steroids)-Reference-Cited by-同舟云学术

Steroidal C-21 heteroaryl thioethers. Part 3: Pregn-4-eno-[3,2-c]pyrazole fused A ring modified steroids as selective glucocorticoid receptor modulators (dissociated steroids)

Published:2012-05 Issue:9 Volume:22 Page:3291-3295
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Biju Purakkattle,Wang Hongwu,Anthes John,McCormick Kevin,Aslanian Robert,Berlin Michael,Bitar Rema,Lim Yeon-Hee,Lee Yoon Joo,Prelusky Daniel,Mcleod Robbie,Jia Yanlin,Fernandez Xiomora,Lieber Gissela,Jimenez Johanna,Eckel Steve,House Aileen,Chapman Richard,Phillips Jonathan

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference15 articles.

1. Steroidal C-21 mercapto derivatives as dissociated steroids: Discovery of an inhaled dissociated steroid

2. Steroidal C-21 heteroaryl thioethers (Part 2): Discovery of orally bioavailable selective glucocorticoid receptor modulators (dissociated steroids)

3. The Three-dimensional Structures of Antagonistic and Agonistic Forms of the Glucocorticoid Receptor Ligand-binding Domain

4. Glide: A New Approach for Rapid, Accurate Docking and Scoring. 1. Method and Assessment of Docking Accuracy

5. Anti-inflammatory Actions of Glucocorticoids: Molecular Mechanisms

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4. Iodine-Promoted Metal-Free Aromatization: Synthesis of Biaryls, Oligop-Phenylenes and A-Ring Modified Steroids;Advanced Synthesis & Catalysis;2015-10-12